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Interactions of quinoline antimalarials with haematin and their effect on ß-haematin formation
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Synthesis and investigation of benzimidazole and carbazole ß-haematin inhibiting scaffolds with antimalarial activity
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Haematin-Quinoline interactions and structure-activity relationships in the antimalarial chloroquine and related compounds
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Interactions of quinoline antimalarial drugs with ferrihaem : structural and kinetic insights into the inhibition of malaria pigment formation
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Kinetics of β-haematin formation in benzoic acid
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Antimalarial Evaluation of Quinoline-triazoleMn(I) and Re(I) PhotoCORMs
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Synthesis of mixed ligand, water soluble square planar platinum (II) complexes and an investigation of their association with haematin and potential to inhibit the formation of synthetic malaria pigment
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Synthesis of 1,4 Dihydropyridines as potential antimalarial chemotype
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Insights into the mechanism of action of quinoline antimalarials against Plasmodium falciparum revealed by novel fluorescent analogues and chemical proteomics
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Single and hybrid antimalarials based on artemisinin, chloroquine and ß-lactams : synthesis, antiplasmodial activity, cytotoxicity and effect of selected artemisinin-chloroquine hybrids on the parasitic endocytosis pathway
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Antimalarial and cysteine protease inhibitor pharmacophores as scaffolds for new antimalarial agents
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Interactions of ferriprotoporphyrin IX with neutral lipids and detergents: insights into their role in β-haematin formation
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Synthesis and evaluation of hybrid compounds based on antimalarial and anticancer pharmacophores
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New aminoquinoline antimalarial cysteine protease inhibitors based on the isatin natural product scaffold
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Antiprotozoal quinolines containing electrophilic moieties
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Curcumin-related hybrid compounds as potential antimalarial agents : design, synthesis, mechanistic investigations, biological evaluation and pharmacokinetic studies
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Elaboration of 4′-Phosphopantetheine Adenylyltransferase inhibitors and Benzoxaboroles as antimalarial agents
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Towards the development of a medium-throughput assay to investigate the kinetics of β-Haematin formation in the presence of divers inhibitors
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Design and synthesis of potential inhibitors of enzymes involved in the biosynthesis and utilisation of mycothiol
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Quinoline-triazole half-sandwich iridium(III) complexes: Synthesis, antiplasmodial activity and preliminary transfer hydrogenation studies
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Bioactive chloroquine-based ligands and their gold complexes as potential novel antimalarial agents
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Synthesis, structure-activity relationship and solubility improvement studies of potential antimalarial and antischistosomal pyrido[1,2-a]benzimidazoles
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Synthesis and Antimalarial evaluation of Gold Thiosemicarbazone Complexes and Polyamine-Thiosemicarbazone Dendrimers
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The design and synthesis of potential acetylcholinesterase inhibitors and NMDA antagonists as neuroprotective agents